Product Name: RU-58841
CAS: 154992-24-2
MF: C17H18F3N3O3
MW: 369.3383
Purity: 99%
BP: 493.6°C at 760 mmHg
FP: 252.3°C
Density: 1.39g/cm3
Grade: Pharmaceutical Grade
Appearance: White Powder
RU58841 is a specific androgen receptor antagonist or a so called anti-androgen. This non steroidal topical androgen antagonist was investigated for therapeutic value in androgenetic alopecia and acne. In studies and clinical trials RU58841 has shown to:
Strongly compete against DHT
Increase cellular replication rate in the matrix cells
Increase cellular proliferation of outer root sheeth cells
Increase hair diameter and hair density
Increase the percentage of hair in the anagen phase
Provide equivalent or better net growth than Finasteride
RU58841 works by binding to the androgen receptor in the hair follicle. Therefore androgens don’t have the chance to bind and start the chain reaction of androgenetic alopecia and begin the so called miniaturization process. It has been demonstrated to interrupt this hair loss message locally so that normal hair growth could continue.
Topical RU58841 has a very short half-life (1 hr) in comparison to the oral ingestion of Finasteride (6 hrs) and Dutasteride (5 weeks!). Moreover, RU58841 does not inhibit DHT production like the latter two products. These facts seem to suggest that there is minimal chance of any serious or permanent side effects, and anecdotal evidence on the forums seems to support that. However, because many people are buying RU58841 from online sometimes unknown and unverified suppliers, there is no guarantee of any kind of safety at all. I am not planning to buy RU58841 online because of safety issues. The product is also quite expensive in comparison to Minoxidil or Finasteride. If you really do wish to buy this product, consult a doctor first.
Side Effects
Despite it being safe in theory, users who have experimented on themselves with RU58841 have reported side effects including:
skin irritation
blurred vision
nausea
dizziness
headaches
reduced libido
erectile dysfunction
Showing posts with label Raw Powder. Show all posts
Showing posts with label Raw Powder. Show all posts
Friday, December 8, 2017
Hair Loss Treatment Powder Minoxidil
Product Name: Minoxidil
Alias: Ioniten,Monoxodyl,Lonolox
CAS: 38304-91-5
EINECS: 253-874-2
MF: C9H15N5O
MW: 209.25
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Hair Loss Treatment
Minoxidil is an antihypertensive vasodilator medication. It also slows hair loss and promotes hair regrowth in some people. Now off-patent, it is available over the counter for the treatment of androgenic alopecia.
Minoxidil, applied topically, is widely used for the treatment of hair loss. It is effective in helping promote hair growth in both males and females with androgenic alopecia.About 40% of men experience hair regrowth after 3-6 months.Minoxidil must be used indefinitely for continued support of existing hair follicles and the maintenance of any experienced hair regrowth.It is the only topical product that is FDA-approved for androgenic hair loss.Treatments usually include a 5% concentration solution that is designed for men, and a 2% concentration solution for women.Minoxidil has been approved for female use by the FDA.
Side Effects
Minoxidil is generally well tolerated, but common side effects include burning or irritation of the eye, itching, redness or irritation at the treated area, as well as unwanted hair growth elsewhere on the body.
Alias: Ioniten,Monoxodyl,Lonolox
CAS: 38304-91-5
EINECS: 253-874-2
MF: C9H15N5O
MW: 209.25
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Hair Loss Treatment
Minoxidil is an antihypertensive vasodilator medication. It also slows hair loss and promotes hair regrowth in some people. Now off-patent, it is available over the counter for the treatment of androgenic alopecia.
Minoxidil, applied topically, is widely used for the treatment of hair loss. It is effective in helping promote hair growth in both males and females with androgenic alopecia.About 40% of men experience hair regrowth after 3-6 months.Minoxidil must be used indefinitely for continued support of existing hair follicles and the maintenance of any experienced hair regrowth.It is the only topical product that is FDA-approved for androgenic hair loss.Treatments usually include a 5% concentration solution that is designed for men, and a 2% concentration solution for women.Minoxidil has been approved for female use by the FDA.
Side Effects
Minoxidil is generally well tolerated, but common side effects include burning or irritation of the eye, itching, redness or irritation at the treated area, as well as unwanted hair growth elsewhere on the body.
Hair Loss Treatment Powder Finasteride
Product Name: Finasteride
Alias: Proscar,Propecia,Fincompared Toteride
CAS: 98319-26-7
MF: C23H36N2O2
MW: 372.55
Purity: 99.68%
Grade: Pharmaceutical Grade
Appearance: White Powder
Treatment Of Enlarged Prostate Gland
Finasteride (Proscar) is a very potent type II 5a-reductase inhibitor, which prevents conversion of testosterone to dihydrotestosterone (DHT). DHT is a sex hormone. In addition, it is used for treatment of benign prostatic hyperplasia (BPH), which is the enlargement of the prostate.
Finasteride inhibits 4a-reductase, and as mentioned, will prevent testosterone conversion to DHT. Studies have shown it will reduce serum DHT levels by about 65-70%, and prostate DHT levels, by up to 90%. By blocking DHT production, finasteride reduces androgen activity on the scalp; and in the prostate reduces prostate volume, which improves BPH, and reduces risk of prostate cancer.
Prevent Hair Loss
Bodybuilders will want to inhibit this conversion as much as possible to preserve hair loss, which is why finasteride is used. This is especially true when using DHT derivative anabolic steroids. Finasteride does a good job at keeping existing hair, and in almost half of men it will help grow more hair.
Finasteride is used to treat male pattern hair loss (androgenetic alopecia) in men only.Treatment provides about 30% improvement in hair loss after six months of treatment, and effectiveness only persists as long as the drug is taken.Clinical studies suggest that, with Finasteride 1 mg/day, continuously taking it for 3 months or slightly long , users can have their hair regrow, after 1 year if continuous treatment, hair growth rate is up to 48%.
Finasteride Dosage
Bodybuilders will dose Finasteride at 1mg per day to preserve hair. This is usually done during their DHT cycles.
Alias: Proscar,Propecia,Fincompared Toteride
CAS: 98319-26-7
MF: C23H36N2O2
MW: 372.55
Purity: 99.68%
Grade: Pharmaceutical Grade
Appearance: White Powder
Treatment Of Enlarged Prostate Gland
Finasteride (Proscar) is a very potent type II 5a-reductase inhibitor, which prevents conversion of testosterone to dihydrotestosterone (DHT). DHT is a sex hormone. In addition, it is used for treatment of benign prostatic hyperplasia (BPH), which is the enlargement of the prostate.
Finasteride inhibits 4a-reductase, and as mentioned, will prevent testosterone conversion to DHT. Studies have shown it will reduce serum DHT levels by about 65-70%, and prostate DHT levels, by up to 90%. By blocking DHT production, finasteride reduces androgen activity on the scalp; and in the prostate reduces prostate volume, which improves BPH, and reduces risk of prostate cancer.
Prevent Hair Loss
Bodybuilders will want to inhibit this conversion as much as possible to preserve hair loss, which is why finasteride is used. This is especially true when using DHT derivative anabolic steroids. Finasteride does a good job at keeping existing hair, and in almost half of men it will help grow more hair.
Finasteride is used to treat male pattern hair loss (androgenetic alopecia) in men only.Treatment provides about 30% improvement in hair loss after six months of treatment, and effectiveness only persists as long as the drug is taken.Clinical studies suggest that, with Finasteride 1 mg/day, continuously taking it for 3 months or slightly long , users can have their hair regrow, after 1 year if continuous treatment, hair growth rate is up to 48%.
Finasteride Dosage
Bodybuilders will dose Finasteride at 1mg per day to preserve hair. This is usually done during their DHT cycles.
Weight Loss Powder T4
Product Name: T4
Alias: levothyroxine,thyroid hormone,L-Thyroxine sodium salt,Levothyroxine Sodium
CAS: 25416-65-3
EINECS: 200-221-4
MF: C15H10I4NNaO4
MW: 798.85
Purity:98%
Appearance: White Powder
Grade: Pharmaceutical Grade
Treatment for Hypercholesterolemia
Levothyroxine or L-thyroxine is a synthetic thyroid hormone that is chemically identical to thyroxine (T4), which is naturally secreted by the follicular cells of the thyroid gland. It is used to treat thyroid hormone deficiency, and occasionally to prevent the recurrence of thyroid cancer. Like its naturally secreted counterpart, levothyroxine is a chiral compound in the L-form. The related drug dextrothyroxine (D-thyroxine) was used in the past as a treatment for hypercholesterolemia (elevated cholesterol levels) but was withdrawn due to cardiac side effects.
Levothyroxine is typically used to treat hypothyroidism, and is the treatment of choice for patients with hypothyroidism, who often require lifelong thyroid hormone therapy. It may also be used to treat goiter via its ability to lower thyroid-stimulating hormone (TSH), a hormone that is considered goiter-inducing. Levothyroxine is also used as interventional therapy in patients with nodular thyroid disease or thyroid cancer to suppress thyroid-stimulating hormone (TSH) secretion.
Fat Loss
Thyroid hormone controls the rate of metabolism. When the thyroid is under active, all body processes slow down and symptoms such as weight gain, fatigue, and decreased body temperature are experienced. Through supplementation of thyroid hormones, basal metabolic rate will be increased.
Thyroid hormones are essential to proper development of all cells in body. These hormones allow for the body to become more sensitive to all other hormones, in turn making them more effective. Thyroid hormones also regulate macronutrient (protein, fat and carbohydrate) metabolism, therefore increasing protein synthesis and ultimately energy. This allows for the body to burn more calories and use them more sufficiently. For this reason, thyroid hormones are commonly used as fat-loss drugs.
Usage and Dosage
Users discovered T3 to be a better choice over T4 when using Thyroid drugs during Cyclic Ketogenic Diets.
T4 must be used in much higher doses to be as effective as T3. Subjects found they needed to use a dosage of 300 mcg/day to achieve the same results as 25-100 mcg/day of T3 (Cytomel).
Alias: levothyroxine,thyroid hormone,L-Thyroxine sodium salt,Levothyroxine Sodium
CAS: 25416-65-3
EINECS: 200-221-4
MF: C15H10I4NNaO4
MW: 798.85
Purity:98%
Appearance: White Powder
Grade: Pharmaceutical Grade
Treatment for Hypercholesterolemia
Levothyroxine or L-thyroxine is a synthetic thyroid hormone that is chemically identical to thyroxine (T4), which is naturally secreted by the follicular cells of the thyroid gland. It is used to treat thyroid hormone deficiency, and occasionally to prevent the recurrence of thyroid cancer. Like its naturally secreted counterpart, levothyroxine is a chiral compound in the L-form. The related drug dextrothyroxine (D-thyroxine) was used in the past as a treatment for hypercholesterolemia (elevated cholesterol levels) but was withdrawn due to cardiac side effects.
Levothyroxine is typically used to treat hypothyroidism, and is the treatment of choice for patients with hypothyroidism, who often require lifelong thyroid hormone therapy. It may also be used to treat goiter via its ability to lower thyroid-stimulating hormone (TSH), a hormone that is considered goiter-inducing. Levothyroxine is also used as interventional therapy in patients with nodular thyroid disease or thyroid cancer to suppress thyroid-stimulating hormone (TSH) secretion.
Fat Loss
Thyroid hormone controls the rate of metabolism. When the thyroid is under active, all body processes slow down and symptoms such as weight gain, fatigue, and decreased body temperature are experienced. Through supplementation of thyroid hormones, basal metabolic rate will be increased.
Thyroid hormones are essential to proper development of all cells in body. These hormones allow for the body to become more sensitive to all other hormones, in turn making them more effective. Thyroid hormones also regulate macronutrient (protein, fat and carbohydrate) metabolism, therefore increasing protein synthesis and ultimately energy. This allows for the body to burn more calories and use them more sufficiently. For this reason, thyroid hormones are commonly used as fat-loss drugs.
Usage and Dosage
Users discovered T3 to be a better choice over T4 when using Thyroid drugs during Cyclic Ketogenic Diets.
T4 must be used in much higher doses to be as effective as T3. Subjects found they needed to use a dosage of 300 mcg/day to achieve the same results as 25-100 mcg/day of T3 (Cytomel).
Weight Loss Powder T3
Product Name:T3,Cytomel
Alias: L-thyronine sodium salt,Cytomel T3
CAS NO: 55-06-1
Einecs No: 200-223-5
MF: C15H11I3NNaO4
MW: 672.96
Purity: 98.0%
Appearance: White Powder
Fat Loss
Liothyronine is the most potent form of thyroid hormone. Chemically, it is nearly identical to triiodothyronine (T3). As such, it acts on the body to increase the basal metabolic rate, affect protein synthesis and increase the body's sensitivity to catecholamines (such as adrenaline) by permissiveness. The thyroid hormones are essential to proper development and differentiation of all cells of the human body. These hormones also regulate protein, fat, and carbohydrate metabolism, affecting how human cells use energetic compounds.
T3 is a regulator of the oxidative metabolism of energy. When you take liothyronine sodium it will increase the uptake of nutrients into the mitochondria, which raises activity in the oxidative metabolic pathway. This causes everything to work harder within the organism and makes the body demand more fuel.
T3 in the body is responsible for regulating the uptake of various nutrients into cells and into the mitochondria of those cells in order to effectively become utilized for the production and consumption of energy.The mitochondria of every single cell in the body utilizes carbohydrates (primarily), fat, and even protein for the production of an energy source known as ATP (Adenosine Triphosphate). Through the intake of more T3, this production of ATP will increase, leading to an increased rate of energy consumption in the form of fats,carbohydrates, and protein. Hence, this is why the consumption of too much T3 without the use of anabolic steroids can result in muscle loss.
Bodybuilding
The increase of ATP and metabolic activity leads the body to burn fat. This is why bodybuilders use T3 as a part of their anabolic steroid stacks. Furthermore, T3 is popular among bodybuilders because it can help burn those stubborn 1 to 2% of body fat that won’t come off through just diet and cardio.
Another interesting property of Cytomel is that it can enhance growth hormone (GH) production.
Dosages of T3
In the first approach, the goal is to achieve an ongoing edge in fat loss or to help maintain a near-personally-ideal body composition. In this approach, T3 dosing is very low, preferably 12.5 mcg/day but in some cases as much as 25 mcg/day. At the lower end of this range, typically thyroid testing will show no detectable suppression even with prolonged use. At the higher end, moderate suppression is sometimes seen, but results are superior to when T3 is not taken, and the suppression reverses rapidly upon discontinuing T3 use.
In the second approach, the goal is to achieve a quite substantial increase in rate of fat loss, at the known cost of inducing thyroid suppression. Most preferably the dosage is about 50 mcg/day, but in some instances can be as high as 75 mcg/day. Such use is preferably not ongoing, but only for a limited period of time such as 8-12 weeks, though there’s no exact requirement for timeframe.
Alias: L-thyronine sodium salt,Cytomel T3
CAS NO: 55-06-1
Einecs No: 200-223-5
MF: C15H11I3NNaO4
MW: 672.96
Purity: 98.0%
Appearance: White Powder
Fat Loss
Liothyronine is the most potent form of thyroid hormone. Chemically, it is nearly identical to triiodothyronine (T3). As such, it acts on the body to increase the basal metabolic rate, affect protein synthesis and increase the body's sensitivity to catecholamines (such as adrenaline) by permissiveness. The thyroid hormones are essential to proper development and differentiation of all cells of the human body. These hormones also regulate protein, fat, and carbohydrate metabolism, affecting how human cells use energetic compounds.
T3 is a regulator of the oxidative metabolism of energy. When you take liothyronine sodium it will increase the uptake of nutrients into the mitochondria, which raises activity in the oxidative metabolic pathway. This causes everything to work harder within the organism and makes the body demand more fuel.
T3 in the body is responsible for regulating the uptake of various nutrients into cells and into the mitochondria of those cells in order to effectively become utilized for the production and consumption of energy.The mitochondria of every single cell in the body utilizes carbohydrates (primarily), fat, and even protein for the production of an energy source known as ATP (Adenosine Triphosphate). Through the intake of more T3, this production of ATP will increase, leading to an increased rate of energy consumption in the form of fats,carbohydrates, and protein. Hence, this is why the consumption of too much T3 without the use of anabolic steroids can result in muscle loss.
Bodybuilding
The increase of ATP and metabolic activity leads the body to burn fat. This is why bodybuilders use T3 as a part of their anabolic steroid stacks. Furthermore, T3 is popular among bodybuilders because it can help burn those stubborn 1 to 2% of body fat that won’t come off through just diet and cardio.
Another interesting property of Cytomel is that it can enhance growth hormone (GH) production.
Dosages of T3
In the first approach, the goal is to achieve an ongoing edge in fat loss or to help maintain a near-personally-ideal body composition. In this approach, T3 dosing is very low, preferably 12.5 mcg/day but in some cases as much as 25 mcg/day. At the lower end of this range, typically thyroid testing will show no detectable suppression even with prolonged use. At the higher end, moderate suppression is sometimes seen, but results are superior to when T3 is not taken, and the suppression reverses rapidly upon discontinuing T3 use.
In the second approach, the goal is to achieve a quite substantial increase in rate of fat loss, at the known cost of inducing thyroid suppression. Most preferably the dosage is about 50 mcg/day, but in some instances can be as high as 75 mcg/day. Such use is preferably not ongoing, but only for a limited period of time such as 8-12 weeks, though there’s no exact requirement for timeframe.
Weight Loss Powder Theobromine
Product Name: Theobromine
Alias: Teobromin,Theominal,Theoxalvose,Riddovydrin,Diurobromine Theobromine
CAS: 83-67-0
EINECS: 201-494-2
MF: C7H8N4O2
MW: 180.16
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Theobromine, formerly known as xantheose, is a bitter alkaloid of the cacao plant, with the chemical formula C7H8N4O2. It is classified as a xanthine alkaloid, which also includes the similar compounds theophylline. The compounds differ in their degree of methylation.
Health Benefits Of Theobromine
Theobromine has a similar effect than caffeine, but about 10 times weaker. Theobromine has diuretic, stimulant and relaxing effects. Theobromine can lower the blood pressure because it can to dilate blood vessels.
Theobromine has stimulant properties, similar to caffeine. Unlike caffeine theobromine does not affect the central nervous system.
Theobromine can also relax bronchi muscles in the lungs. Theobromine can be used as cough medicine. Studies indicate that theobromine acts on the vagus nerve, which runs from the lungs to the brain.
Weight Loss
Theobromine is a mild stimulant and diuretic. Both of these properties can aid weight loss by giving you a little energy boost for physical activity and helping you shed water weight. Theobromine can also help suppress your appetite. Theobromine can be said to promote weight loss in a variety of different ways including vasodilatation, diuresis and the ability to increase energy although most of these seem to be indirect.
Use
In modern medicine, theobromine is used as a vasodilator (a blood vessel widener), a diuretic (urination aid), and heart stimulant. Theobromine increases urine production. Because of this diuretic effect, and its ability to dilate blood vessels, theobromine has been used to treat high blood pressure.
Alias: Teobromin,Theominal,Theoxalvose,Riddovydrin,Diurobromine Theobromine
CAS: 83-67-0
EINECS: 201-494-2
MF: C7H8N4O2
MW: 180.16
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Theobromine, formerly known as xantheose, is a bitter alkaloid of the cacao plant, with the chemical formula C7H8N4O2. It is classified as a xanthine alkaloid, which also includes the similar compounds theophylline. The compounds differ in their degree of methylation.
Health Benefits Of Theobromine
Theobromine has a similar effect than caffeine, but about 10 times weaker. Theobromine has diuretic, stimulant and relaxing effects. Theobromine can lower the blood pressure because it can to dilate blood vessels.
Theobromine has stimulant properties, similar to caffeine. Unlike caffeine theobromine does not affect the central nervous system.
Theobromine can also relax bronchi muscles in the lungs. Theobromine can be used as cough medicine. Studies indicate that theobromine acts on the vagus nerve, which runs from the lungs to the brain.
Weight Loss
Theobromine is a mild stimulant and diuretic. Both of these properties can aid weight loss by giving you a little energy boost for physical activity and helping you shed water weight. Theobromine can also help suppress your appetite. Theobromine can be said to promote weight loss in a variety of different ways including vasodilatation, diuresis and the ability to increase energy although most of these seem to be indirect.
Use
In modern medicine, theobromine is used as a vasodilator (a blood vessel widener), a diuretic (urination aid), and heart stimulant. Theobromine increases urine production. Because of this diuretic effect, and its ability to dilate blood vessels, theobromine has been used to treat high blood pressure.
Weight Loss Powder Telmisartan
Product Name: Telmisartan
Alias: Micardis
CAS: 144701-48-4
MF: C33H30N4O2
MW: 514.62
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Telmisartan (Micardis) is an oral prescription medication most commonly used to treat hypertension, including mild hypertension where blood pressure is only moderately elevated or borderline. If choosing to self-medicate for mild hypertension or borderline high blood pressure, telmisartan is an excellent or even best choice.
As elevated blood pressure is often an undesired side effect of anabolic steroid cycles and can even limit use of androgens, this use of telmisartan is already enough to make the drug of value to many.
However, telmisartan also has an entirely different category of use, due to having quite a number of other interesting properties which can be valuable in some instances.
Benefits can include improvement to fat loss, endurance, insulin sensitivity, reduction of risk of atherosclerosis, stroke, and of heart attack, and possible benefit to brain health. In some cases mood or energy can be improved as well.
When To Use Telmisartan
If blood pressure needs to be moderated, I'd certainly consider using telmisartan. If there is no such need, factors that could suggest its use include interest in reducing visceral fat, of improving impaired insulin sensitivity, of reducing risk of atherosclerosis, or depending on personal interest, of possibly improving brain health and function.
Reasons not to use telmisartan could include unwillingness to accept the risk of possible side effects, or unwillingness to shift the balance of fat loss towards visceral fat loss versus subcutaneous fat loss. In general, if dieting and training achieve only the same bodyfat percentage despite the positive effects of telmisartan, appearance could be smoother due to the same amount of bodyfat being present but with less of it stored as unhealthful visceral fat. On the other hand, if taking advantage of improved loss of visceral fat with telmisartan to achieve a lower bodyfat percentage, then there's no smoothness penalty. However, when aiming for contest condition there's a certain amount of fat that the body must retain: theoretically, reducing visceral fat in this case might force retention of a greater amount of subcutaneous fat. So I wouldn't advise telmisartan use in the last few weeks before a bodybuilding contest.
How To Use Telmisartan
To reduce risk of atherosclerosis, cardiovascular disease, or stroke where risk is only moderate in the first place, I suggest a dose from 20 to 40 mg taken orally once per day. Dosing would be the same where the interest is slowing loss of brain function with age, or potentially improving brain function.
For possible improvement in fat loss, particularly of visceral fat, or improvement of endurance I suggest dosing of 80-160 mg/day. Starting dose, however, generally should be only 40 mg/day until tolerance is assessed.
While it's not required and telmisartan users in general do not do so, when using this drug I suggest supplementing with oleuropein 200-400 mg/day and Vitamin D 5000 IU/day. These are to reduce or perhaps eliminate two activities of telmisartan that I would not consider desirable for physique or performance enhancement, though they add to its medical use.
Telmisartan should not be used in combination with a diuretic, and I would avoid allowing severe dehydration while using this drug.
Blood pressure should be monitored while using telmisartan. Typically, any decrease of blood pressure is simply to healthful levels or more-nearly healthful levels, and those who do not have high blood pressure see no decrease with telmisartan. Still, there can be exceptions, so this should be watched.
Lastly, I would cycle telmisartan use rather than use it continuously. There's no proof of what cycling method might be optimal, but for example I'd suggest being "off" about as many weeks per year as "on" as a minimum. This is not because of proven problem, but simply because I expect the benefits can be fully or nearly fully realized with this amount of use, and where any of the changes to gene expression or receptor blocking might be adverse in the individual case rather than beneficial, this will then be no more than half the time.
Alias: Micardis
CAS: 144701-48-4
MF: C33H30N4O2
MW: 514.62
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Telmisartan (Micardis) is an oral prescription medication most commonly used to treat hypertension, including mild hypertension where blood pressure is only moderately elevated or borderline. If choosing to self-medicate for mild hypertension or borderline high blood pressure, telmisartan is an excellent or even best choice.
As elevated blood pressure is often an undesired side effect of anabolic steroid cycles and can even limit use of androgens, this use of telmisartan is already enough to make the drug of value to many.
However, telmisartan also has an entirely different category of use, due to having quite a number of other interesting properties which can be valuable in some instances.
Benefits can include improvement to fat loss, endurance, insulin sensitivity, reduction of risk of atherosclerosis, stroke, and of heart attack, and possible benefit to brain health. In some cases mood or energy can be improved as well.
When To Use Telmisartan
If blood pressure needs to be moderated, I'd certainly consider using telmisartan. If there is no such need, factors that could suggest its use include interest in reducing visceral fat, of improving impaired insulin sensitivity, of reducing risk of atherosclerosis, or depending on personal interest, of possibly improving brain health and function.
Reasons not to use telmisartan could include unwillingness to accept the risk of possible side effects, or unwillingness to shift the balance of fat loss towards visceral fat loss versus subcutaneous fat loss. In general, if dieting and training achieve only the same bodyfat percentage despite the positive effects of telmisartan, appearance could be smoother due to the same amount of bodyfat being present but with less of it stored as unhealthful visceral fat. On the other hand, if taking advantage of improved loss of visceral fat with telmisartan to achieve a lower bodyfat percentage, then there's no smoothness penalty. However, when aiming for contest condition there's a certain amount of fat that the body must retain: theoretically, reducing visceral fat in this case might force retention of a greater amount of subcutaneous fat. So I wouldn't advise telmisartan use in the last few weeks before a bodybuilding contest.
How To Use Telmisartan
To reduce risk of atherosclerosis, cardiovascular disease, or stroke where risk is only moderate in the first place, I suggest a dose from 20 to 40 mg taken orally once per day. Dosing would be the same where the interest is slowing loss of brain function with age, or potentially improving brain function.
For possible improvement in fat loss, particularly of visceral fat, or improvement of endurance I suggest dosing of 80-160 mg/day. Starting dose, however, generally should be only 40 mg/day until tolerance is assessed.
While it's not required and telmisartan users in general do not do so, when using this drug I suggest supplementing with oleuropein 200-400 mg/day and Vitamin D 5000 IU/day. These are to reduce or perhaps eliminate two activities of telmisartan that I would not consider desirable for physique or performance enhancement, though they add to its medical use.
Telmisartan should not be used in combination with a diuretic, and I would avoid allowing severe dehydration while using this drug.
Blood pressure should be monitored while using telmisartan. Typically, any decrease of blood pressure is simply to healthful levels or more-nearly healthful levels, and those who do not have high blood pressure see no decrease with telmisartan. Still, there can be exceptions, so this should be watched.
Lastly, I would cycle telmisartan use rather than use it continuously. There's no proof of what cycling method might be optimal, but for example I'd suggest being "off" about as many weeks per year as "on" as a minimum. This is not because of proven problem, but simply because I expect the benefits can be fully or nearly fully realized with this amount of use, and where any of the changes to gene expression or receptor blocking might be adverse in the individual case rather than beneficial, this will then be no more than half the time.
Weight Loss Powder Synephrine
Product Name: Synephrine
Alias: Oxedrine
CAS: 94-07-5
EINECS: 202-300-9
MF: C9H13NO2
MW: 167.205
Assay: 98%
Grade: Pharmaceutical Grade
Appearance: White Powder
Application Scope
Synephrine is one of the adrenergic amines that stimulates the beta-3 receptors with minimal impact on the other receptor sites. This functions to increase the metabolic rate without affecting heart rate or blood pressure. Synephrine releases adrenaline and noradrenaline only in the beta-3 receptor sites (mostly adipose tissue and the liver). Stimulation of the beta-3 receptor sites elicits the breakdown of lipolysis (fat).Synephrine is used to activate the adrenaline system without the stimulatory effect posed by ephedra-based products.
In application of traditional Chinese medical science, Synephrine is used to dispel bloating and a lump in the abdomen and phlegm, and to cureedema, constipation, gastroptosis, prolapse of uterus and rectocele.Anti- tumour, prevent osteoporosis, reduce cholesterin and protect heart.Nerve protection and prevent diseases of degeneration ofnerve.Relieve menopausal symptoms of women, improve bone metabolism and protect cardiovascular system, etc.
Fat Loss
Synephrine is a stimulant, similar to caffeine and ephedrine. It is thought to have similar effects in terms of providing an energy boost, suppressing appetite and increasing metabolic rate leading to the burning or more calories. It is used as a safer alternative to Ma Huang, synephrine is theorized to stimulate fat metabolism without the negative cardiovascular side effects experienced by some people with Ma Huang.
The most likely explanation for weight loss effects attributed to citrus aurantium (synephrine) supplements is the stimulant like effects of the alkaloids. Although this effect is likely to be somewhat less dramatic that effects induced by Ma Huang (ephedra - also known as Sida Cordifolia), users can expect variable effects including reduced appetite and heightened feelings of energy (similar to caffeine)... both of which are likely to result in weight loss.
Synephrine Dosage
Take about 5-20mg of synephrine two to three times per day, having one of those doses 30-60 minutes prior to workouts.
Alias: Oxedrine
CAS: 94-07-5
EINECS: 202-300-9
MF: C9H13NO2
MW: 167.205
Assay: 98%
Grade: Pharmaceutical Grade
Appearance: White Powder
Application Scope
Synephrine is one of the adrenergic amines that stimulates the beta-3 receptors with minimal impact on the other receptor sites. This functions to increase the metabolic rate without affecting heart rate or blood pressure. Synephrine releases adrenaline and noradrenaline only in the beta-3 receptor sites (mostly adipose tissue and the liver). Stimulation of the beta-3 receptor sites elicits the breakdown of lipolysis (fat).Synephrine is used to activate the adrenaline system without the stimulatory effect posed by ephedra-based products.
In application of traditional Chinese medical science, Synephrine is used to dispel bloating and a lump in the abdomen and phlegm, and to cureedema, constipation, gastroptosis, prolapse of uterus and rectocele.Anti- tumour, prevent osteoporosis, reduce cholesterin and protect heart.Nerve protection and prevent diseases of degeneration ofnerve.Relieve menopausal symptoms of women, improve bone metabolism and protect cardiovascular system, etc.
Fat Loss
Synephrine is a stimulant, similar to caffeine and ephedrine. It is thought to have similar effects in terms of providing an energy boost, suppressing appetite and increasing metabolic rate leading to the burning or more calories. It is used as a safer alternative to Ma Huang, synephrine is theorized to stimulate fat metabolism without the negative cardiovascular side effects experienced by some people with Ma Huang.
The most likely explanation for weight loss effects attributed to citrus aurantium (synephrine) supplements is the stimulant like effects of the alkaloids. Although this effect is likely to be somewhat less dramatic that effects induced by Ma Huang (ephedra - also known as Sida Cordifolia), users can expect variable effects including reduced appetite and heightened feelings of energy (similar to caffeine)... both of which are likely to result in weight loss.
Synephrine Dosage
Take about 5-20mg of synephrine two to three times per day, having one of those doses 30-60 minutes prior to workouts.
Weight Loss Powder Rimonabant
Product Name: Rimonabant
Alias: Acomplia,Zimulti,Rimonabdomining Exercisesish
CAS: 168273-06-1
MF: C22H21Cl3N4O
MW: 463.79
Purity: 99.5%
Grade: Pharmaceutical Grade
Appearance: White Powder
Weight Loss
Rimonabant (trade name Acomplia) is an anorectic antiobesity drug that has been withdrawn from the market due to potentially serious side effects.Rimonabant is an inverse agonist for the cannabinoid receptor CB1.It has also been shown to be a μ-opioid receptor antagonist (possibly the contributing factor in its reported dysphoric qualities).Its main effect is reduction in appetite.Rimonabant works by blocking the cannabinoid receptors in the brain. This is designed to lower your food cravings in between meals and prevent you from munching on snacks when your body doesn't truly need food. The recommended dosage is only a single pill each day before breakfast.
The Rimonabant is a very great weight loss powders in nowadays markets ,and its purity is very high ,the contents is for 99% ;especially for smoker and is also for patients with cardiovascular diseases.
Application
1)Obesity,weight loss
2)Smoking cessation
3)Addiction behaviors
4)Short-term memory
5)Blockage of cannabis effects
Alias: Acomplia,Zimulti,Rimonabdomining Exercisesish
CAS: 168273-06-1
MF: C22H21Cl3N4O
MW: 463.79
Purity: 99.5%
Grade: Pharmaceutical Grade
Appearance: White Powder
Weight Loss
Rimonabant (trade name Acomplia) is an anorectic antiobesity drug that has been withdrawn from the market due to potentially serious side effects.Rimonabant is an inverse agonist for the cannabinoid receptor CB1.It has also been shown to be a μ-opioid receptor antagonist (possibly the contributing factor in its reported dysphoric qualities).Its main effect is reduction in appetite.Rimonabant works by blocking the cannabinoid receptors in the brain. This is designed to lower your food cravings in between meals and prevent you from munching on snacks when your body doesn't truly need food. The recommended dosage is only a single pill each day before breakfast.
The Rimonabant is a very great weight loss powders in nowadays markets ,and its purity is very high ,the contents is for 99% ;especially for smoker and is also for patients with cardiovascular diseases.
Application
1)Obesity,weight loss
2)Smoking cessation
3)Addiction behaviors
4)Short-term memory
5)Blockage of cannabis effects
Weight Loss Powder Orlistat
Product Name: Orlistat
CAS: 96829-58-2
MF: C29H53NO5
MW: 495.73
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Fat Loss Mechanism
Orlistat is a drug that promotes loss of weight by preventing the digestion and absorption of fat in food. In the intestine, an enzyme called lipase (produced primarily by the pancreas) breaks apart fat in food so that it can be absorbed into the body. Orlistat blocks the action of lipase and thereby prevents the breakup and absorption of fat. Orlistat blocks absorption of about 25% of the fat in a meal. The unabsorbed fat is excreted in the stool.
This medication is used along with a doctor-approved reduced-calorie diet, exercise, and behavior modification program to help significantly overweight (obese) persons lose weight. Taking orlistat can also help prevent you from regaining the weight you have lost. Losing weight and keeping it off can reduce the many health risks that obesity causes, including heart disease, diabetes, high blood pressure, some forms of cancer, certain breathing problems, and a shorter life span.
Dietary fats need to be broken down into smaller pieces before the body can absorb them. Orlistat works by blocking the enzyme that breaks down fats in your diet. This undigested fat then passes out of your body in your bowel movement. Orlistat does not block the absorption of calories from sugar and other non-fat foods, so you still need to restrict your total intake of calories.
Fat Loss Effect
Orlistat is used for the treatment of obesity. The amount of weight loss achieved with orlistat varies. In one-year clinical trials, between 35.5% and 54.8% of subjects achieved a 5% or greater decrease in body mass, although not all of this mass was necessarily fat. Between 16.4% and 24.8% achieved at least a 10% decrease in body fat.After orlistat was stopped, a significant number of subjects regained weight-up to 35% of the weight they had lost.
The incidence of type 2 diabetes in an obese population over four years is decreased with orlistat (6.2%) compared to placebo (9.0%).Long-term use of orlistat also leads to a modest reduction in blood pressure (mean reductions of 2.5 and 1.9 mmHg in systolic and diastolic blood pressure respectively).
Orlistat Dosage
Orlistat is usually taken 3 times a day during every meal containing fat. The average dosage is a 120mg per day. Due to the fact that Xenical may decrease the absorption of vitamins and it is useful to take a multivitamin once a day at bedtime. While taking this drug bodybuilders and athletes should follow their diet, medication, and exercise routines very closely.
CAS: 96829-58-2
MF: C29H53NO5
MW: 495.73
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Fat Loss Mechanism
Orlistat is a drug that promotes loss of weight by preventing the digestion and absorption of fat in food. In the intestine, an enzyme called lipase (produced primarily by the pancreas) breaks apart fat in food so that it can be absorbed into the body. Orlistat blocks the action of lipase and thereby prevents the breakup and absorption of fat. Orlistat blocks absorption of about 25% of the fat in a meal. The unabsorbed fat is excreted in the stool.
This medication is used along with a doctor-approved reduced-calorie diet, exercise, and behavior modification program to help significantly overweight (obese) persons lose weight. Taking orlistat can also help prevent you from regaining the weight you have lost. Losing weight and keeping it off can reduce the many health risks that obesity causes, including heart disease, diabetes, high blood pressure, some forms of cancer, certain breathing problems, and a shorter life span.
Dietary fats need to be broken down into smaller pieces before the body can absorb them. Orlistat works by blocking the enzyme that breaks down fats in your diet. This undigested fat then passes out of your body in your bowel movement. Orlistat does not block the absorption of calories from sugar and other non-fat foods, so you still need to restrict your total intake of calories.
Fat Loss Effect
Orlistat is used for the treatment of obesity. The amount of weight loss achieved with orlistat varies. In one-year clinical trials, between 35.5% and 54.8% of subjects achieved a 5% or greater decrease in body mass, although not all of this mass was necessarily fat. Between 16.4% and 24.8% achieved at least a 10% decrease in body fat.After orlistat was stopped, a significant number of subjects regained weight-up to 35% of the weight they had lost.
The incidence of type 2 diabetes in an obese population over four years is decreased with orlistat (6.2%) compared to placebo (9.0%).Long-term use of orlistat also leads to a modest reduction in blood pressure (mean reductions of 2.5 and 1.9 mmHg in systolic and diastolic blood pressure respectively).
Orlistat Dosage
Orlistat is usually taken 3 times a day during every meal containing fat. The average dosage is a 120mg per day. Due to the fact that Xenical may decrease the absorption of vitamins and it is useful to take a multivitamin once a day at bedtime. While taking this drug bodybuilders and athletes should follow their diet, medication, and exercise routines very closely.
Weight Loss Powder L-Carnitine
Product Name: L-Carnitine
Alias: Vitamin BT,L-Ca Greatrnitine,L-Ctheirrnitine
CAS: 541-15-1
EINECS: 208-768-0
MF: C7H15NO3
MW: 161.20
Appearance: White Powder
Melting Point: 200 dec.
Description
L-Carnitine is a natural, vitamin-like nutrient wich plays an important role inhuman metabolism. It is essential in the utilization of fatty acids and in transporting metabolic energy.
Carnitine (carnitine) is an essential, non-toxic, natural nutrient that helps burn fat for fuel. Because deficiencies have been linked to a profound impairment of muscle function, there has been great interest in studying carnitine supplementation. Over the past decade, my research, as well as countless others, has shed light on carnitine's role in metabolism, performance and overall health.
Carnitine Burns Body Fat
Carnitine has an essential role in transporting fat into mitochondria (the furnace of the cell). Therefore, carnitine has been marketed as a fat burning supplement.Carnitine is a substance that helps the body turn fat into energy. Your body makes it in the liver and kidneys and stores it in the skeletal muscles, heart, brain, and sperm.
Usually, your body can make all the carnitine it needs. Some people, however, may not have enough carnitine because their bodies cannot make enough or can't transport it into tissues so it can be used. Some other conditions, such as angina or intermittent claudication, can also cause low levels of carnitine in the body, as can some medications.
Carnitine has been proposed as a treatment for many conditions because it acts as an antioxidant. Antioxidants fight harmful particles in the body known as free radicals, which damage cells and tamper with DNA. Antioxidants can neutralize free radicals and may reduce or help prevent some of the damage they cause.
Alias: Vitamin BT,L-Ca Greatrnitine,L-Ctheirrnitine
CAS: 541-15-1
EINECS: 208-768-0
MF: C7H15NO3
MW: 161.20
Appearance: White Powder
Melting Point: 200 dec.
Description
L-Carnitine is a natural, vitamin-like nutrient wich plays an important role inhuman metabolism. It is essential in the utilization of fatty acids and in transporting metabolic energy.
Carnitine (carnitine) is an essential, non-toxic, natural nutrient that helps burn fat for fuel. Because deficiencies have been linked to a profound impairment of muscle function, there has been great interest in studying carnitine supplementation. Over the past decade, my research, as well as countless others, has shed light on carnitine's role in metabolism, performance and overall health.
Carnitine Burns Body Fat
Carnitine has an essential role in transporting fat into mitochondria (the furnace of the cell). Therefore, carnitine has been marketed as a fat burning supplement.Carnitine is a substance that helps the body turn fat into energy. Your body makes it in the liver and kidneys and stores it in the skeletal muscles, heart, brain, and sperm.
Usually, your body can make all the carnitine it needs. Some people, however, may not have enough carnitine because their bodies cannot make enough or can't transport it into tissues so it can be used. Some other conditions, such as angina or intermittent claudication, can also cause low levels of carnitine in the body, as can some medications.
Carnitine has been proposed as a treatment for many conditions because it acts as an antioxidant. Antioxidants fight harmful particles in the body known as free radicals, which damage cells and tamper with DNA. Antioxidants can neutralize free radicals and may reduce or help prevent some of the damage they cause.
Weight Loss Powder DNP
Product Name: DNP
Alias: Sodium DNP;Sodium 2,4-dinitrophenolate;Sodium 2,4-dinitrophenoxide
CAS: 1011-73-0
EINECS: 213-786-7
MF: C6H3N2NaO5
MW: 206.0882
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: Yellow Crystalline
BP: 312.1°C at 760 mmHg
FP: 142.8°C
DNP is an extremely powerful fat burning drug. There is no compound on earth that can burn fat at the rate of DNP; however, to say it is beyond dangerous is almost an understatement. DNP is so dangerous it can in fact kill you. No one can deny the fat loss power held by this compound is truly tremendous, but when we consider the risk there are very few if any we can recommend it too.
Effects of DNP
The effects of DNP are very simple and very straightforward, tremendous fat loss and loss of total bodyweight. So powerful, the effects of DNP can result in a full pound of body fat loss per day. Note we said a full pound of body fat, not merely weight but actual pure body fat. That is truly amazing and could easily result in twenty plus pounds of fat loss in only a few weeks, not to mention any other weight lost, i.e. water weight.
That's it, pure fat loss, rapid and tremendous fat loss represents the full effects of DNP. The compound carries no additional traits that could be potentially desired by any human being. While sometimes labeled as a performance enhancing drug DNP carries no anabolic properties. The compound will not help the individual build muscle mass or enhance strength. The individual will not see his athletic performance enhanced; in fact, many would see it diminished as DNP can be extremely draining on energy levels. Further, due to the tremendous increase in body temperature, when we look at the side effects of DNP we will find extreme activity must be avoided when using the compound.
When looking at the effects of DNP in a performance setting, many are often curious about its fat loss power compared to other more commonly used medications. The two most commonly used fat loss aids in performance enhancement circles are undoubtedly Clenbuterol and Cytomel (T3), and both are highly effective. However, while we cannot recommend DNP and while both Clen and T3 are far safer, we cannot deny the truth. DNP is far more powerful and will lead to greater and more dramatic fat loss than both Clenbuterol and Cytomel combined. This is simply the truth; however, both Clenbuterol and Cytomel can easily be used without severe or even fatal consequences, but we cannot say the same for DNP.
Side Effects of DNP
The most common side effects of DNP use include dramatic insomnia, nausea and extreme sweating. When we refer to extreme sweating, a more accurate way to describe it would be sweating profusely. Many who have used DNP have reported ruining their mattress during periods of use due to the sweating being so intense. DNP is also well-known for causing cataracts, which in many cases ultimately leads to the individual going blind.
DNP can also have a strong, negative impact on white blood cell count by reducing the total count severely. This can have a disastrous effect on the individual's immune system. You will be far more susceptible to viruses and infections when using DNP. It is also very common for those who use DNP to fall into a coma, which can very easily lead to an untimely death.
Alias: Sodium DNP;Sodium 2,4-dinitrophenolate;Sodium 2,4-dinitrophenoxide
CAS: 1011-73-0
EINECS: 213-786-7
MF: C6H3N2NaO5
MW: 206.0882
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: Yellow Crystalline
BP: 312.1°C at 760 mmHg
FP: 142.8°C
DNP is an extremely powerful fat burning drug. There is no compound on earth that can burn fat at the rate of DNP; however, to say it is beyond dangerous is almost an understatement. DNP is so dangerous it can in fact kill you. No one can deny the fat loss power held by this compound is truly tremendous, but when we consider the risk there are very few if any we can recommend it too.
Effects of DNP
The effects of DNP are very simple and very straightforward, tremendous fat loss and loss of total bodyweight. So powerful, the effects of DNP can result in a full pound of body fat loss per day. Note we said a full pound of body fat, not merely weight but actual pure body fat. That is truly amazing and could easily result in twenty plus pounds of fat loss in only a few weeks, not to mention any other weight lost, i.e. water weight.
That's it, pure fat loss, rapid and tremendous fat loss represents the full effects of DNP. The compound carries no additional traits that could be potentially desired by any human being. While sometimes labeled as a performance enhancing drug DNP carries no anabolic properties. The compound will not help the individual build muscle mass or enhance strength. The individual will not see his athletic performance enhanced; in fact, many would see it diminished as DNP can be extremely draining on energy levels. Further, due to the tremendous increase in body temperature, when we look at the side effects of DNP we will find extreme activity must be avoided when using the compound.
When looking at the effects of DNP in a performance setting, many are often curious about its fat loss power compared to other more commonly used medications. The two most commonly used fat loss aids in performance enhancement circles are undoubtedly Clenbuterol and Cytomel (T3), and both are highly effective. However, while we cannot recommend DNP and while both Clen and T3 are far safer, we cannot deny the truth. DNP is far more powerful and will lead to greater and more dramatic fat loss than both Clenbuterol and Cytomel combined. This is simply the truth; however, both Clenbuterol and Cytomel can easily be used without severe or even fatal consequences, but we cannot say the same for DNP.
Side Effects of DNP
The most common side effects of DNP use include dramatic insomnia, nausea and extreme sweating. When we refer to extreme sweating, a more accurate way to describe it would be sweating profusely. Many who have used DNP have reported ruining their mattress during periods of use due to the sweating being so intense. DNP is also well-known for causing cataracts, which in many cases ultimately leads to the individual going blind.
DNP can also have a strong, negative impact on white blood cell count by reducing the total count severely. This can have a disastrous effect on the individual's immune system. You will be far more susceptible to viruses and infections when using DNP. It is also very common for those who use DNP to fall into a coma, which can very easily lead to an untimely death.
Weight Loss Powder DMAA
Product Name: 1,3-Dimethylpentylamine HCL
Alias: DMAA,Dimethylamylamine,Methylhexamine,Methylhexanamine
CAS: 13803-74-2
MF: C7H18ClN
MW: 151.68
Grade: Pharmaceutical Grade
Appearance: White Powder
Methylhexanamine is synthesized by reacting 4-methylhexanone-2 with hydroxylamine, which converts the 4-methylhexanone-2 to 4-methylhexanone-2 oxime, which is reduced with hydrogen by means of a catalyst; the resulting methylhexanamine can be purified by distillation.
Fat Loss
A large number of supplements focusing on fat loss and workout energy (thermogenic or general-purpose stimulants) now use the ingredient in concert with other substances such as caffeine, a combination similar to the combination of ephedrine and caffeine.
Methylhexanamine is an indirect sympathomimetic drug that constricts blood vessels and thus has effects on the heart, lungs, and reproductive organs it also causes bronchodilation, inhibits peristalsis in the intestines, and has diuretic effects.Most studies have been done on pharmacological effects when the drug is inhaled; our understanding of what methylhexanamine does when taken orally are mostly based on extrapolating from the activities of similar compounds.Today, dimethylamylamine is sold as a dietary supplement used for attention deficit-hyperactive disorder (ADHD), weight loss, improving athletic performance, and body building.
Athletes and bodybuilders are constantly persuing lean body mass.When it comes to sports performance and building,some turn to dietary and sports improving supplements to boost their athletic performance or lose body fat. One such supplement ingredient called methylhexamamine or DMAA is advertised for this objective and is currently the topic of some controversy.
How Does DMAA Work?
DMAA has stimulant results significantly like caffeine. Individuals who take it experience more energized and have better mental focus without any the jitteriness that many people experience when they drink an excessive amount of caffeine. At exactly the same time, DMAA causes constriction of blood vessels and dilation of bronchioles in the lungs. It's also an appetite suppressant and may cause weight loss in some people.
Using And Dosage
A typical starting dose of 1,3-DMAA is in the 10-20mg range and eventually reaching up to 40-60mg a day, there is no actual evidence to support this dosage range but it seems to be the standard dosages range for supplemental 1,3-DMAA on the market.
Alias: DMAA,Dimethylamylamine,Methylhexamine,Methylhexanamine
CAS: 13803-74-2
MF: C7H18ClN
MW: 151.68
Grade: Pharmaceutical Grade
Appearance: White Powder
Methylhexanamine is synthesized by reacting 4-methylhexanone-2 with hydroxylamine, which converts the 4-methylhexanone-2 to 4-methylhexanone-2 oxime, which is reduced with hydrogen by means of a catalyst; the resulting methylhexanamine can be purified by distillation.
Fat Loss
A large number of supplements focusing on fat loss and workout energy (thermogenic or general-purpose stimulants) now use the ingredient in concert with other substances such as caffeine, a combination similar to the combination of ephedrine and caffeine.
Methylhexanamine is an indirect sympathomimetic drug that constricts blood vessels and thus has effects on the heart, lungs, and reproductive organs it also causes bronchodilation, inhibits peristalsis in the intestines, and has diuretic effects.Most studies have been done on pharmacological effects when the drug is inhaled; our understanding of what methylhexanamine does when taken orally are mostly based on extrapolating from the activities of similar compounds.Today, dimethylamylamine is sold as a dietary supplement used for attention deficit-hyperactive disorder (ADHD), weight loss, improving athletic performance, and body building.
Athletes and bodybuilders are constantly persuing lean body mass.When it comes to sports performance and building,some turn to dietary and sports improving supplements to boost their athletic performance or lose body fat. One such supplement ingredient called methylhexamamine or DMAA is advertised for this objective and is currently the topic of some controversy.
How Does DMAA Work?
DMAA has stimulant results significantly like caffeine. Individuals who take it experience more energized and have better mental focus without any the jitteriness that many people experience when they drink an excessive amount of caffeine. At exactly the same time, DMAA causes constriction of blood vessels and dilation of bronchioles in the lungs. It's also an appetite suppressant and may cause weight loss in some people.
Using And Dosage
A typical starting dose of 1,3-DMAA is in the 10-20mg range and eventually reaching up to 40-60mg a day, there is no actual evidence to support this dosage range but it seems to be the standard dosages range for supplemental 1,3-DMAA on the market.
Tuesday, December 5, 2017
Sex Enhancement Powder Yohimbine HCL
Product Name: Yohimbine HCL
Alias: Corynine,Aphrodine,Yohimbe HCl,Yohimbe,Yohimbine,Yoh,Yohimar,Testomar,Erex
CAS: 65-19-0
EINECS: 200-600-4
MF: C21H26N2O3HCL
MW: 390.91
Purity: 98%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Better Sex, Better Erections
Yohimbine HCl has shown to rapidly increase the Libido of both men and women and its properties as an aphrodisiac are well known throughout the scientific world. Yohimbine HCl increases the sex drive of men and is even used to treat hypoactive sexual desire disorder (under active libido) in women.
Its most pronounced sexual effect appears to be in its treatment of Erectile Dysfunction in men and has shown to even increase penile girth (the width of the male penis). Through its effect on minor corpus cavernosum smooth muscle relaxation, the vasodilatation caused increases blood flow to the penis exponentially. Continual use of Yohimbine HCl is required to achieve these results as it cannot be achieved through casual or one time usage.
Energy, Appetite Suppression, & Weight Loss
Numerous studies have shown Yohimbe in all its forms will increase energy, has shown to increase the heart rate in sedentary individuals, and is well known as a powerful fat loss compound. Through its appetite suppressing functions and metabolism increasing functions, this one-two punch has shown to be a catalyst for powerful weight loss in both men and women alike.
The biggest mistake made by users of this prescription grade element is when it is taken with food. Yohimbe in all its forms must be taken on an empty stomach in between meals in order to achieve maximum effectiveness. Food and certain vitamins will nullify the effects of Yohimbine HCl and this is even present in some supplements which contain this powerful element.
The weight loss benefits of it can be quite powerful and extreme when taken in its proper dosing and in its purest form.
Yohimbine Dosage & Administration
First off, Yohimbine HCl must NOT be taken with food or vitamin supplements of any kind. It must be taken by itself on an empty stomach in between meals or in a fasted state when you first wake up in the morning. It also is best to spread dosing throughout the day as this also helps with its appetite suppressing effects which will help maximize your weight loss when taking it.
Dosing: The minimum dosing is set at 5 mg per day, with 2.5 mg taken 2 times per day on an empty stomach in between meals as described above. Do not take with any other supplement. Wait at least 20-30 minutes until you eat after administration.
Maximum Results: In order to achieve the maximum effects when taking this supplement, the following dosing guidelines should be met.
Dosages of 0.2mg/kg bodyweight have been successfully used to increase fat burning without significant implications on cardiovascular parameters like heart rate and blood pressure. This results in a dosage of: 14 mg for a 150lb person, 18 mg for a 200lb person, and 22 mg for a 250lb person.
Alias: Corynine,Aphrodine,Yohimbe HCl,Yohimbe,Yohimbine,Yoh,Yohimar,Testomar,Erex
CAS: 65-19-0
EINECS: 200-600-4
MF: C21H26N2O3HCL
MW: 390.91
Purity: 98%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Better Sex, Better Erections
Yohimbine HCl has shown to rapidly increase the Libido of both men and women and its properties as an aphrodisiac are well known throughout the scientific world. Yohimbine HCl increases the sex drive of men and is even used to treat hypoactive sexual desire disorder (under active libido) in women.
Its most pronounced sexual effect appears to be in its treatment of Erectile Dysfunction in men and has shown to even increase penile girth (the width of the male penis). Through its effect on minor corpus cavernosum smooth muscle relaxation, the vasodilatation caused increases blood flow to the penis exponentially. Continual use of Yohimbine HCl is required to achieve these results as it cannot be achieved through casual or one time usage.
Energy, Appetite Suppression, & Weight Loss
Numerous studies have shown Yohimbe in all its forms will increase energy, has shown to increase the heart rate in sedentary individuals, and is well known as a powerful fat loss compound. Through its appetite suppressing functions and metabolism increasing functions, this one-two punch has shown to be a catalyst for powerful weight loss in both men and women alike.
The biggest mistake made by users of this prescription grade element is when it is taken with food. Yohimbe in all its forms must be taken on an empty stomach in between meals in order to achieve maximum effectiveness. Food and certain vitamins will nullify the effects of Yohimbine HCl and this is even present in some supplements which contain this powerful element.
The weight loss benefits of it can be quite powerful and extreme when taken in its proper dosing and in its purest form.
Yohimbine Dosage & Administration
First off, Yohimbine HCl must NOT be taken with food or vitamin supplements of any kind. It must be taken by itself on an empty stomach in between meals or in a fasted state when you first wake up in the morning. It also is best to spread dosing throughout the day as this also helps with its appetite suppressing effects which will help maximize your weight loss when taking it.
Dosing: The minimum dosing is set at 5 mg per day, with 2.5 mg taken 2 times per day on an empty stomach in between meals as described above. Do not take with any other supplement. Wait at least 20-30 minutes until you eat after administration.
Maximum Results: In order to achieve the maximum effects when taking this supplement, the following dosing guidelines should be met.
Dosages of 0.2mg/kg bodyweight have been successfully used to increase fat burning without significant implications on cardiovascular parameters like heart rate and blood pressure. This results in a dosage of: 14 mg for a 150lb person, 18 mg for a 200lb person, and 22 mg for a 250lb person.
Sex Enhancement Powder Vardenafil
Product Name: Vardenafil
Alias: Levitra,Fardenafil,Vardenafil HCL
CAS: 224785-91-5
MF: C23H32N6O4S
MW: 525.06
Assay: 98%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Vardenafil Effect
Vardenafil is a PDE5 inhibitor used for treating erectile dysfunction. Vardenafil's indications and contra-indications are the same as with other PDE5 inhibitors; it is closely related in function to Sildenafil citrate (Viagra) and Tadalafil (Cialis). The difference between the Vardenafil molecule and Sildenafil citrate is that a nitrogen atom has different position and the change of Sildenafil's piperazine ring methyl group to an ethyl group. Tadalafil is structurally different from both Sildenafil and Vardenafil. Vardenafil's relatively short effective time is comparable to but somewhat longer than Sildenafil's.
Further, Vardenafil lengthens QT interval. Therefore it should not be taken by men taking other medications that affect the QT interval (such as Amiodarone).
Vardenafil Dosage
Patients taking Levitra are usually started on a 10 mg dose, which they take no more than once daily, about one hour before sexual activity. It can take as little as 30 minutes for Levitra to work in some patients. Like with Viagra, Levitra dosages are adjusted depending on a person's reaction, with doctors generally decreasing doses to to 2.5 mg or increasing them to no more than 20 mg once a day.
Vardenafil, as with all PDE5 inhibitors, should not be used by men taking nitrate medications, because combining them with Vardenafil might provoke potentially life-threatening hypotension (low blood pressure).
Vardenafil Side Effects
Facial flushing (reddening), headaches, stomach upset, diarrhea, flu like symptoms and nausea. Vardenafil also may cause chest pain, low blood pressure, blurred vision and changes in color vision, abnormal ejaculation and priapism (painful erection).
Alias: Levitra,Fardenafil,Vardenafil HCL
CAS: 224785-91-5
MF: C23H32N6O4S
MW: 525.06
Assay: 98%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Vardenafil Effect
Vardenafil is a PDE5 inhibitor used for treating erectile dysfunction. Vardenafil's indications and contra-indications are the same as with other PDE5 inhibitors; it is closely related in function to Sildenafil citrate (Viagra) and Tadalafil (Cialis). The difference between the Vardenafil molecule and Sildenafil citrate is that a nitrogen atom has different position and the change of Sildenafil's piperazine ring methyl group to an ethyl group. Tadalafil is structurally different from both Sildenafil and Vardenafil. Vardenafil's relatively short effective time is comparable to but somewhat longer than Sildenafil's.
Further, Vardenafil lengthens QT interval. Therefore it should not be taken by men taking other medications that affect the QT interval (such as Amiodarone).
Vardenafil Dosage
Patients taking Levitra are usually started on a 10 mg dose, which they take no more than once daily, about one hour before sexual activity. It can take as little as 30 minutes for Levitra to work in some patients. Like with Viagra, Levitra dosages are adjusted depending on a person's reaction, with doctors generally decreasing doses to to 2.5 mg or increasing them to no more than 20 mg once a day.
Vardenafil, as with all PDE5 inhibitors, should not be used by men taking nitrate medications, because combining them with Vardenafil might provoke potentially life-threatening hypotension (low blood pressure).
Vardenafil Side Effects
Facial flushing (reddening), headaches, stomach upset, diarrhea, flu like symptoms and nausea. Vardenafil also may cause chest pain, low blood pressure, blurred vision and changes in color vision, abnormal ejaculation and priapism (painful erection).
Sex Enhancement Powder Tadalafil
Product Name: Tadalafil
Alias: Calais,Ciingis,Cingais,Cialisr,Chinacialisr,Cialis
CAS: 171596-29-5
MF: C22H19N3O4
MW: 389.341
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Tadalafil Effect
Like its predecessor Viagra, Tadalifil is used to treat erectile dysfunction in men. One of the more embarrassing side effects of post-cycle-therapy is the decreased libido caused by the sudden absence of exaggerated testosterone levels in the body, often leading to ED. If you cann't get it up after your cycle, get the pill.
Tadalifil, a phosphodiesterase type 5 inhibitor, is used to treat erectile dysfunction (ED) and decreased libido in males. Cialis works by aiding relaxation of blood vessels and increasing blood flow in the penis during sexual arousal, resulting in improved erectile function. Cialis is much longer lasting than Viagra. Effects can be felt anywhere between 36-48 hours.
Tadalafil improves erectile function significantly, possibly increase testosterone through increased sexual activity, and is very safe.Cialis was also linked to increased testosterone levels in a one month study where testosterone levels were found to be significantly higher at the end of the month, due to increased sexual activity.
Applications
1.It is used for treatment of decreased libido caused by the sudden absence of exaggerated testosterone levels in the body.
2.How ironic. Some of the compounds which can be used to make men more physically attractive to women (Deca, Tren, etc…)
3.Cialis is useful for these occasions…or during PCT when sexual dysfunction may occur.
Tadalifil Side Effects
There are limited side effects associated with its use. The most common side effects are headache, upset stomach, back pain, and muscle aches, and usually subside with in a few hours.
Alias: Calais,Ciingis,Cingais,Cialisr,Chinacialisr,Cialis
CAS: 171596-29-5
MF: C22H19N3O4
MW: 389.341
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Tadalafil Effect
Like its predecessor Viagra, Tadalifil is used to treat erectile dysfunction in men. One of the more embarrassing side effects of post-cycle-therapy is the decreased libido caused by the sudden absence of exaggerated testosterone levels in the body, often leading to ED. If you cann't get it up after your cycle, get the pill.
Tadalifil, a phosphodiesterase type 5 inhibitor, is used to treat erectile dysfunction (ED) and decreased libido in males. Cialis works by aiding relaxation of blood vessels and increasing blood flow in the penis during sexual arousal, resulting in improved erectile function. Cialis is much longer lasting than Viagra. Effects can be felt anywhere between 36-48 hours.
Tadalafil improves erectile function significantly, possibly increase testosterone through increased sexual activity, and is very safe.Cialis was also linked to increased testosterone levels in a one month study where testosterone levels were found to be significantly higher at the end of the month, due to increased sexual activity.
Applications
1.It is used for treatment of decreased libido caused by the sudden absence of exaggerated testosterone levels in the body.
2.How ironic. Some of the compounds which can be used to make men more physically attractive to women (Deca, Tren, etc…)
3.Cialis is useful for these occasions…or during PCT when sexual dysfunction may occur.
Tadalifil Side Effects
There are limited side effects associated with its use. The most common side effects are headache, upset stomach, back pain, and muscle aches, and usually subside with in a few hours.
Sex Enhancement Powder Sildenafil Citrate
Product Name: Sildenafil Citrate
Synonyms: Viagra,Revatio,Sildenafil Citrdined,Sildenafil Citrgot,Sildenafil Citringested
CAS: 171599-83-0
MF: C28H38N6O11S
MW: 666.7
Assay: 98.8%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Sildenafil Citrate Effect
Sildenafil Citrate, sold as Viagra, Revatio and under various other trade names, is a drug used to treat erectile dysfunction and pulmonary arterial hypertension (PAH). It acts by inhibiting cGMP-specific phosphodiesterase type 5 (PDE5), an enzyme that promotes degradation of cGMP, which regulates blood flow in the penis.
The primary indication of sildenafil is treatment of erectile dysfunction (inability to sustain a satisfactory erection to complete intercourse). Its use is now standard treatment for erectile dysfunction in all settings, including diabetes.
Medical Uses
1)Sexual dysfunction
2)Pulmonary hypertension
3)Antidepressant-associated sexual dysfunction
4)Altitude sickness
Sildenafil Dosage
Viagra: for erectile dysfunction, comes in blue, diamond-shaped pills, in doses of 25, 50, or 100 milligrams. The patient takes a maximum of one pill in a 24-hour period, between 30 minutes to 1 hour before sexual intercourse.
Revatio: for pulmonary arterial hypertension, comes in white, round, film-coated tablets. Patients take one 20 mg Revatio tablet three times a day.
Synonyms: Viagra,Revatio,Sildenafil Citrdined,Sildenafil Citrgot,Sildenafil Citringested
CAS: 171599-83-0
MF: C28H38N6O11S
MW: 666.7
Assay: 98.8%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Sildenafil Citrate Effect
Sildenafil Citrate, sold as Viagra, Revatio and under various other trade names, is a drug used to treat erectile dysfunction and pulmonary arterial hypertension (PAH). It acts by inhibiting cGMP-specific phosphodiesterase type 5 (PDE5), an enzyme that promotes degradation of cGMP, which regulates blood flow in the penis.
The primary indication of sildenafil is treatment of erectile dysfunction (inability to sustain a satisfactory erection to complete intercourse). Its use is now standard treatment for erectile dysfunction in all settings, including diabetes.
Medical Uses
1)Sexual dysfunction
2)Pulmonary hypertension
3)Antidepressant-associated sexual dysfunction
4)Altitude sickness
Sildenafil Dosage
Viagra: for erectile dysfunction, comes in blue, diamond-shaped pills, in doses of 25, 50, or 100 milligrams. The patient takes a maximum of one pill in a 24-hour period, between 30 minutes to 1 hour before sexual intercourse.
Revatio: for pulmonary arterial hypertension, comes in white, round, film-coated tablets. Patients take one 20 mg Revatio tablet three times a day.
Sex Enhancement Powder Flibanserin
Product Name: Flibanserin
CAS: 167933-07-5
MF: C20H21F3N4O
MW: 390.40
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Flibanserin, sold under the trade name Addyi, is a medication approved for the treatment of pre-menopausal women with hypoactive sexual desire disorder (HSDD).The medication increases the number of satisfying sexual events per month by about one half to one over placebo from a starting point of about two to three.
Flibanserin is used for hypoactive sexual desire disorder among women. Those receiving flibanserin report that the average number of times they had "satisfying sexual events" rose from 2.8 to 4.5 times a month. However, women receiving placebo reported also an increase of "satisfying sexual events" from 2.7 to 3.7 times a month. Evaluation of the overall improvement of their condition and whether the benefit was meaningful to the women, showed a significantly higher rate of a meaningful benefit in the flibanserin-treated people versus the placebo group.The onset of the flibanserin effect was seen from the first timepoint measured after 4 weeks of treatment and maintained throughout the treatment period.
The effectiveness of flibanserin was evaluated in three phase 3 clinical trials. Each of the three trials had two co-primary endpoints, one for satisfying sexual events (SSEs) and the other for sexual desire. Each of the 3 trials also had a secondary endpoint that measured distress related to sexual desire.
All three trials showed that flibanserin produced a statistically significant increase in the number of SSEs and reduced distress related to sexual desire.
The first two trials used an electronic diary to measure sexual desire, and did not find a statistically significant increase relative to women treated with a placebo. These two trials also measured sexual desire using the Female Sexual Function index (FSFI) as a secondary endpoint, and a statistically significant increase was observed using this latter measure. The FSFI was used as the co-primary endpoint for sexual desire in the third trial, and again showed a statistically significant increase.
CAS: 167933-07-5
MF: C20H21F3N4O
MW: 390.40
Purity: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Flibanserin, sold under the trade name Addyi, is a medication approved for the treatment of pre-menopausal women with hypoactive sexual desire disorder (HSDD).The medication increases the number of satisfying sexual events per month by about one half to one over placebo from a starting point of about two to three.
Flibanserin is used for hypoactive sexual desire disorder among women. Those receiving flibanserin report that the average number of times they had "satisfying sexual events" rose from 2.8 to 4.5 times a month. However, women receiving placebo reported also an increase of "satisfying sexual events" from 2.7 to 3.7 times a month. Evaluation of the overall improvement of their condition and whether the benefit was meaningful to the women, showed a significantly higher rate of a meaningful benefit in the flibanserin-treated people versus the placebo group.The onset of the flibanserin effect was seen from the first timepoint measured after 4 weeks of treatment and maintained throughout the treatment period.
The effectiveness of flibanserin was evaluated in three phase 3 clinical trials. Each of the three trials had two co-primary endpoints, one for satisfying sexual events (SSEs) and the other for sexual desire. Each of the 3 trials also had a secondary endpoint that measured distress related to sexual desire.
All three trials showed that flibanserin produced a statistically significant increase in the number of SSEs and reduced distress related to sexual desire.
The first two trials used an electronic diary to measure sexual desire, and did not find a statistically significant increase relative to women treated with a placebo. These two trials also measured sexual desire using the Female Sexual Function index (FSFI) as a secondary endpoint, and a statistically significant increase was observed using this latter measure. The FSFI was used as the co-primary endpoint for sexual desire in the third trial, and again showed a statistically significant increase.
Antiestrogen Powder Raloxifene HCL
Product Name: Raloxifene HCL
CAS: 82640-04-8
MF: C28H28ClNO4S
MW: 510.05
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: Light Yellow Powder
Usage: Pharmaceutical Raw Materials
Raloxifene HCL is an oral selective estrogen receptor modulator (SERM) that has estrogenic actions on bone and anti-estrogenic actions on the uterus and breast. It is used in the prevention of osteoporosis in postmenopausal women and to reduce the risk of invasive breast cancer in postmenopausal women with osteoporosis and in postmenopausal women at high risk for invasive breast cancer.
This drug is different from hormones (including estrogens and progestins). It works by acting like estrogen (as a selective estrogen receptor modulator or SERM) in some parts of the body. Raloxifene helps to preserve bone mass, but it does not affect the breast and uterus like estrogen or relieve symptoms of menopause such as hot flashes.
Raloxifene is indicated for the treatment and prevention of osteoporosis in postmenopausal women. It is also used for reduction of risk and treatment of invasive breast cancer, and it also reduces breast density.For either osteoporosis treatment or prevention, supplemental calcium and/or vitamin D should be added to the diet if daily intake is inadequate.
Raloxifene is used to prevent and treat bone loss (osteoporosis) in women after menopause. Maintaining strong bones by slowing bone loss helps to reduce the risk of fractures.
Raloxifene may also lower the chance of getting a certain type of breast cancer (invasive) in women after menopause.
CAS: 82640-04-8
MF: C28H28ClNO4S
MW: 510.05
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: Light Yellow Powder
Usage: Pharmaceutical Raw Materials
Raloxifene HCL is an oral selective estrogen receptor modulator (SERM) that has estrogenic actions on bone and anti-estrogenic actions on the uterus and breast. It is used in the prevention of osteoporosis in postmenopausal women and to reduce the risk of invasive breast cancer in postmenopausal women with osteoporosis and in postmenopausal women at high risk for invasive breast cancer.
This drug is different from hormones (including estrogens and progestins). It works by acting like estrogen (as a selective estrogen receptor modulator or SERM) in some parts of the body. Raloxifene helps to preserve bone mass, but it does not affect the breast and uterus like estrogen or relieve symptoms of menopause such as hot flashes.
Raloxifene is indicated for the treatment and prevention of osteoporosis in postmenopausal women. It is also used for reduction of risk and treatment of invasive breast cancer, and it also reduces breast density.For either osteoporosis treatment or prevention, supplemental calcium and/or vitamin D should be added to the diet if daily intake is inadequate.
Raloxifene is used to prevent and treat bone loss (osteoporosis) in women after menopause. Maintaining strong bones by slowing bone loss helps to reduce the risk of fractures.
Raloxifene may also lower the chance of getting a certain type of breast cancer (invasive) in women after menopause.
Antiestrogen Powder Toremifene Citrate
Product Name: Toremifene Citrate
Synonyms: Fareston
CAS: 89778-27-8
MF: C26H28ClNO.C6H8O7
MW: 598.09
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Melting Point: 158-164 dec.
Boiling Point: 535.1 dec. at 760 mmHg
Density: 1.045g/cm3
Refractive Index: 1,416-1,418
Toremifene Citrate Effect
Toremifene citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. Licensed in the United States under the brand name Fareston, toremifene citrate is FDA-approved for use in advanced (metastatic) breast cancer. It is also being evaluated for prevention of prostate cancer under the brand name Acapodene.
It has already been covered that Toremifene is a SERM, and serves to block Estrogen at various receptor sites in certain tissues within the body (breast tissue in particular). As a layman explanation, Toremifene pretends to be a 'fake' Estrogen that occupies Estrogen receptors within breast tissue. With these receptors occupied by Toremifene, real Estrogen cannot perform their jobs there. Toremifene does not reduce total blood plasma levels of Estrogen. In addition to being antagonistic to Estrogen receptors in breast tissue, it is also antagonistic to Estrogen at the hypothalamus gland (this essentially 'tricks' the hypothalamus into thinking there is little or no circulating Estrogen levels in the body, causing it to increase its manufacture of Testosterone so that it can utilize aromatization to restore these levels.
Toremifene Citrate exerts its effects by antagonizing the estrogen receptor in some tissues, and agonizing it in others. In this way, certain estrogenic pathways are activated and others are blockaded. It seems to exert estrogenic effects on blood lipids, reducing LDL and total cholesterol, as well as estrogenic effects on bone, improving density. It would also appear to exert anti-estrogenic effects in breast tissue, displacing the traditional effects of estrogen, effectively helping prevent breast cancer in postmenopausal women.
Fareston Administration
In the fight against breast cancer, standard Fareston doses will normally be 60mg per day. The total duration of use is unpredictable and will be based on patient need. It's not uncommon for treatment to last a year or two and then AI's to be added if needed. Once the cancer is in remission, compounds like Fareston are commonly used to support the improved state.
For the anabolic steroid user combating gynecomastia, standard Fareston doses will fall in the 30-60mg per day range and will work very well for most men. If this is not enough protection, while you could try increasing the dose your best bet would be to move to AI use. You will find Fareston works very well in combating gynecomastia due to the use of any testosterone, Dianabol and Anadrol. You will also find it works well with Equipoise and Deca Durabolin. However, as Deca Durabolin is also a progestin, men who are very sensitive to that hormone may need an AI. The same can be said of the Trenbolone hormone. Trenbolone does not aromatize, but it is a progestin. Further, the use of an aromatizing steroid with a compound like Trenbolone can increase the risk of gynecomastia in some men. While many will not need gynecomastia protection due to progestins and will get by with SERM's to combat aromatase, some sensitive men will need an AI. Regardless, if Fareston works for you it will cover the entire breadth of the cycle from start to finish.
Synonyms: Fareston
CAS: 89778-27-8
MF: C26H28ClNO.C6H8O7
MW: 598.09
Assay: 99%
Grade: Pharmaceutical Grade
Appearance: White Powder
Usage: Pharmaceutical Raw Materials
Melting Point: 158-164 dec.
Boiling Point: 535.1 dec. at 760 mmHg
Density: 1.045g/cm3
Refractive Index: 1,416-1,418
Toremifene Citrate Effect
Toremifene citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. Licensed in the United States under the brand name Fareston, toremifene citrate is FDA-approved for use in advanced (metastatic) breast cancer. It is also being evaluated for prevention of prostate cancer under the brand name Acapodene.
It has already been covered that Toremifene is a SERM, and serves to block Estrogen at various receptor sites in certain tissues within the body (breast tissue in particular). As a layman explanation, Toremifene pretends to be a 'fake' Estrogen that occupies Estrogen receptors within breast tissue. With these receptors occupied by Toremifene, real Estrogen cannot perform their jobs there. Toremifene does not reduce total blood plasma levels of Estrogen. In addition to being antagonistic to Estrogen receptors in breast tissue, it is also antagonistic to Estrogen at the hypothalamus gland (this essentially 'tricks' the hypothalamus into thinking there is little or no circulating Estrogen levels in the body, causing it to increase its manufacture of Testosterone so that it can utilize aromatization to restore these levels.
Toremifene Citrate exerts its effects by antagonizing the estrogen receptor in some tissues, and agonizing it in others. In this way, certain estrogenic pathways are activated and others are blockaded. It seems to exert estrogenic effects on blood lipids, reducing LDL and total cholesterol, as well as estrogenic effects on bone, improving density. It would also appear to exert anti-estrogenic effects in breast tissue, displacing the traditional effects of estrogen, effectively helping prevent breast cancer in postmenopausal women.
Fareston Administration
In the fight against breast cancer, standard Fareston doses will normally be 60mg per day. The total duration of use is unpredictable and will be based on patient need. It's not uncommon for treatment to last a year or two and then AI's to be added if needed. Once the cancer is in remission, compounds like Fareston are commonly used to support the improved state.
For the anabolic steroid user combating gynecomastia, standard Fareston doses will fall in the 30-60mg per day range and will work very well for most men. If this is not enough protection, while you could try increasing the dose your best bet would be to move to AI use. You will find Fareston works very well in combating gynecomastia due to the use of any testosterone, Dianabol and Anadrol. You will also find it works well with Equipoise and Deca Durabolin. However, as Deca Durabolin is also a progestin, men who are very sensitive to that hormone may need an AI. The same can be said of the Trenbolone hormone. Trenbolone does not aromatize, but it is a progestin. Further, the use of an aromatizing steroid with a compound like Trenbolone can increase the risk of gynecomastia in some men. While many will not need gynecomastia protection due to progestins and will get by with SERM's to combat aromatase, some sensitive men will need an AI. Regardless, if Fareston works for you it will cover the entire breadth of the cycle from start to finish.
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